Advanced Peptide Synthesis

Specialized synthesis formats that go beyond routine SPPS—multivalent architectures, conformational constraints, hybrid conjugates, precision handles, and discovery-ready libraries. Use this hub to jump into detailed service pages.

Complex architectures Conformational control Hybrid & conjugates Screening & libraries

Need standard services? See Custom Peptide Synthesis.

Multivalent & Architecture-Controlled Peptides

Topologies that increase epitope density, avidity, or enable site-specific functionalization.

TopologyBranched
Branched Peptide Synthesis

Multi-arm peptides built from a defined branching point to increase functional density or enable multi-epitope formats.

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ImmunologyMAPs
Multiple Antigen Peptides (MAPs)

Dendrimeric constructs that present multiple copies of an epitope without carrier proteins for antibody and vaccine workflows.

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AvidityMultivalent
Multivalent Peptide Synthesis

Peptides engineered to display multiple motifs to improve receptor engagement, potency, or immune recognition.

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DesignCys-selective
Cysteine-Selective Design

Strategic cysteine placement for site-specific conjugation or controlled cyclization while minimizing off-target thiol chemistry.

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Illustration of multivalent and architecture-controlled peptide designs

Representative architectures for branched, MAPs, multivalent, and cysteine-selective peptide designs.

Constrained & Conformationally Controlled Peptides

Formats designed to stabilize bioactive conformations and improve binding specificity or proteolytic stability.

CyclizationCyclic
Cyclic Peptide Synthesis

Cyclic formats (head-to-tail or side-chain) that improve stability and binding by locking peptides into defined geometries.

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ConformationStapled
Stapled Peptide Synthesis

Helix-stabilized peptides using side-chain “staples” to enhance affinity, protease resistance, and functional performance.

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CyclizationMacrocyclic
Macrocyclic Peptide Synthesis

Large cyclic peptides produced via head-to-tail or side-chain cyclization to enhance stability, selectivity, and target engagement.

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CyclizationBicyclic
Bicyclic Peptide Synthesis

Two-ring constrained peptides that increase rigidity and specificity—useful for high-affinity binders and challenging targets.

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StructureHelical
Helical / Constrained Peptide

Conformation-biased designs that stabilize secondary structure (e.g., helix-promoting residues or constraints) for improved activity.

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Stapled peptide (helix stabilization) illustration

Visual: helix stabilization via a side-chain staple.

Hybrid & Bioconjugate Peptides

Peptides combined with lipids, glycans, oligonucleotides, or small molecules to create multifunctional constructs.

GlycoDefined sugars
Glycopeptide Synthesis

Peptides bearing defined carbohydrate moieties for immunology, receptor recognition, and glyco-epitope studies.

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LipidationLipopeptides
Lipopeptide Synthesis

Peptides conjugated to lipid chains to support membrane interaction, delivery strategies, or immune activation.

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ConjugatesOligo
Peptide-Oligonucleotide Conjugates

Hybrid constructs combining peptides with oligonucleotides (DNA/RNA/PNA/PMO) for targeting, delivery, or mechanistic studies.

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HybridSmall molecule
Peptide-Small Molecule Hybrids

Peptides chemically linked to small molecules to add functionality, targeting, or pharmacology to a peptide scaffold.

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Peptide–oligonucleotide and peptide–drug conjugates illustration

Examples of peptide–oligonucleotide and peptide–drug conjugate architectures.

Precision Labeling & Functional Handles

Build in measurement, release, or downstream chemistry with isotope labels, cleavable linkers, and click-ready handles.

Mass specStable isotope
Isotope-Labeled Peptides

Stable isotope incorporation for quantitative LC–MS/MS, pharmacokinetics, or metabolic studies.

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Controlled releaseCleavable
Cleavable Linker Peptides

Peptides with enzyme- or condition-sensitive linkers (pH/redox/protease) for triggered cleavage and payload release.

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BioorthogonalClick-ready
Click Chemistry Peptides

Peptides with bioorthogonal handles for rapid, site-specific conjugation (e.g., azide/alkyne or tetrazine ligations).

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Advanced Design & Discovery Platforms

Formats optimized for screening, mimicry, and immunology tools.

MimicryStability
Peptidomimetics

Peptide-like molecules designed to retain bioactivity while improving stability, permeability, or proteolysis resistance.

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ImmunologyT-cell tools
Custom MHC Peptide Tetramers

Peptide–MHC complexes produced for antigen-specific T-cell detection, immune profiling, and flow cytometry applications.

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LibrariesScreening
Combinatorial Peptide Synthesis

Library-based synthesis generating large collections of related sequences for high-throughput screening and hit discovery.

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CONTACT

Speak to a Peptide Scientist

Share your sequence(s), intended application, purity/scale needs, and any labels or conjugations. We’ll recommend a practical strategy and provide a quote.

Tip: If your project includes multiple sequences (libraries), tell us the count and any shared specifications to speed quoting.

FAQ

Is this page a replacement for peptide modifications?

No. This is an advanced synthesis hub (how peptides are built). Modifications (e.g., labels, PEG, cyclization chemistry) can be separate pages and linked from the relevant services.

How should I request a quote for multiple advanced formats?

Provide sequences (or a spreadsheet), desired purity/scale, required handles (e.g., cysteine, click), and your application. We’ll recommend the most robust build + QC plan.

Do advanced formats affect yield or lead time?

Often, yes. Constrained, hybrid, and library workflows can add steps (special reagents, orthogonal protection, extra QC). We’ll align expectations in the quote.

Can I link each tile to a detail page?

Yes—each card is designed as a gateway. Keep this hub short, and place specs, options, and deeper FAQ content on the linked pages.

Why Choose Bio-Synthesis

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